Caafimaadka, Diyaarinta
"Thiotriazoline": tilmaamaha loo isticmaalo
Ha aad saxiixdo daroogada "Thiotriazoline"? on isticmaalka hage dawadan lagu tilmaami doonaa si faahfaahsan maqaal la joogo. Intaa waxaa dheer, waxaan kuu sheegi doonaa ah oo ku saabsan foomkan, taas oo daroogada gala iibka sheegay, taas oo uu leeyahay tilmaamo, waxyeelo iyo sababo.
Halabuurka ee baakooyinka daroogada iyo foomka fasaxa
In foomka waxa medicament "Thiotriazoline" sii daayo? Tilmaamaha wargalinaya in uu leeyahay tiro ka mid ah noocyada kala duwan. The ugu caansan waa:
- Xalka loogu talagalay duridda iyo faleebo. 1 ml ee wakiilka ka kooban 0,025 Thiotriazoline g. Sidoo kale medicament iyo qaybaha optional qaab biyo la isku duro. daroogada waxaa laga heli karaa 4 ml ampoules (meeleeyay kartoonka).
- "Thiotriazoline" indhaha lagu dhibciyo. By isticmaalka hage noocan oo kale ah waxay ka dhigan tahay waxay bixisaa in 5 ml ka kooban 50 mg daroogada Thiotriazoline, iyo sidoo kale waxyaabaha kale. Daawada waxaa lagu iibiyo dhalooyin caag ah, droppers, meeleeyay kartoon ah.
- kiniinka "Thiotriazoline". Tilmaamaha in foomkan of daroogada waxay bixisaa in ka mid ah kiniinada cadcad ee wareeg ah iyadoo dusha a flat ku jira 100 mg morfoliniymetiltriazoliltioatsetata, ama wax-u Thiotriazoline. Sida qaybaha dheeraad ah medicament ku dhaqmo istaarijka baradho, cellulose mikrokristallin, Hoosaynta miisaanka kelli povidone, milmahayn calcium iyo sucrose. Sida caadiga ah, in xirmo kartoonada ah waxaa ku jira 50 kaniini oo.
pharmacodynamics
Waa maxay daawaynta sida "Thiotriazoline"? Tilmaamaha Isticmaalka dhigayaa in this daroogada antioxidant. Its oolnimada sare waxaa sabab u ah poesie guryaha, antiischemic, immunomodulatory iyo xuub xasilinta.
daawo viewed ka hortagtaa burburinta hepatocytes, kordhinayaan in ay dib u soo kabashada, yaraynaysaa heerka uu dhexgalka dufanka leh, taasoo keentay in caadi of protein, carbohydrate, la egyahay iyo is-dhaafsiga Midabka, iyo yaraynaysaa suurtagalnimada of faafinta galleeyda tsentrolobulyarnyh jirka ah sida beerka. Intaas waxaa sii dheer, daroogada firfircoon hagaajinaysaa faquuqa iyo Avv bile, normalizes ay ka kooban (kiimiko).
The sifooyinka daroogada
Sidee ayaa sifooyinka daroogada "Thiotriazoline"? Tilmaamaha loogu isticmaalo daroogada waxaa looga baahan yahay akhriska. Ka dib oo dhan, ka kaliya ee aad ku baran kartaa oo ku saabsan waxa daroogada loo arkaa hoos u Iscelin of hababka oxidative in wareegga Krebs ah, ilaalinta qasnadda intracellular ATP, iyo sidoo kale kor u hawlgelinta (magdhawga) glycolysis anaerobic ah.
Sidoo kale ogsoonow in ka dib markii walax firfircoon daroogada bilaabmin si aad u bilowdo nidaamka antioxidant, dufanka joogsada geedi socodka oxidative ee meelaha ischaemic ee jirka. Intaa waxaa dheer, daroogada this hagaajinaysaa guryaha (rheology) oo dhiig ah ay sabab u tahay hawshooda u ah ee nidaamka fibrinolytic.
The guryaha poesie of daroogada muujiyey by xaqiiqada ah in qaab-dhismeedka Britain waa udhigo tiotrazolina baaruud, lagu gartaa qaababka lagu qayilo iyo hoos, iyo sidoo kale nitrogen sare, taas oo xidhana lacagta xad dhaaf ah ee atammada hydrogen.
Sidoo kale waa in Waxaan la soco in qayb daroogada firfircoon dhici karta inay xag la egyahay iyo noocyada ogsijiin Waxyeelo. Tan waxa u sabab ah sifooyinka hoos u fahmayaan of group thiol ah. Intaa waxaa dheer, medicament ka hortagtaa formation of noocyada ogsijiin Waxyeelo, falgalka antiradical sida reactivating sida catalase, perodoxida hiddo iyo dismutase superoxide.
Pharmacokinetics
Haddii daawada nuugo "Thiotriazoline"? Waxbarashada dhigayaa in daroogada poluabsorbtsii muddada waa 30 daqiiqo iyo bioavailability - 65.5%.
Ugu badnaan hab-fiirsashada dhiigga waxaa lagu gaarayaa iyada oo 1.4 saacadood ka dib markii maamulka. Isgaarsiinta la borotiinada kama badna 10%.
In u tiro badan, dawada ururayaa in unugyada beerka, wadnaha, xiidanka, beeryarada, iyo kelyihii, iyo yar - xiidmaha yar iyo sambabada. Thiotriazoline inta badan saxarrada kelyaha.
maragga
Haddii ay jiraan leexashooyinkaasi loo xilsaaray karaa kaniiniyada, irbado iyo indhaha lagu dhibciyo "Thiotriazoline"? on isticmaalka noocyadan edbinta muujinaysaa calaamado muujinaya soo socda:
- cirrhosis,
- dhaawaca beerka sun ah, khamri, viral, iyo daroogada (tus, kadib markii la siiyay antibiotics, fayruska daroogada, anti-TB wakiilada iyo anti-buro, piller iyo murugada tricyclic);
- hepatitis viral chronic;
- hepatitis khamriga chronic dhexdhexaad ah hawlaha ugu yar;
- xumaanshaha beerka dufan.
Tilmaamayaasha loo isticmaalo dhibcood:
- cudurada corneal;
- gubasho ama isha dhaawac;
- conjunctivitis viral.
Waa maxay sababta ay weli isticmaalaan daroogada indhaha "Thiotriazoline"? Tilmaamaha (dhibcood laga iibsan karaa farmashiye kasta) ka warrami in daawo this waxaa badanaa loo qoray, waayo, ka hortagga ee isha qalalan, in indhuhu ku daalaan, iyo cudurrada kale ee bararka xubnaha muuqaal ah.
kiniiniyada qiyaasta
Sidee baan u isticmaalaan "Thiotriazoline" kiniin? Buugga waxaa ku jira macluumaad in daroogada waa in la qaato gudaha oo kaliya. Sida caadiga ah, doorataa thiotriazolin 1 ama 2 kaniini oo afar jeer maalintii for 25-30 maalmood.
Muddada aad daawada wakiilka waa in la caddeeyo dhakhtar shakhsiga ku saleysan (ku xiran koorsada iyo adkaanta cudur jira).
Xalka daroogada "Thiotriazoline": tilmaamaha loo isticmaalo
Cirbadaha "Thiotriazoline" samayn intramuscularly ama faleebo. Waxay qiyaasta go'aamiyo dhakhtarka (ku xiran tahay cudurka). Wadnaxanuun myocardial infarction iyo hepatitis daroogada si tartiib ah isku duro intravenously in 2 ml 2-3 jeer maalintii. In cirrhosis medicament waxaa intramuscularly maamulo (2 ml 2-3 jeer maalintii). koorsada daawada waa 60 maalmood.
Indhaha lagu dhibciyo "Thiotriazoline": tilmaamaha loo isticmaalo
Indhaha lagu dhibciyo "Thiotriazoline" Ruhbaaniyad gelin koleyga conjunctival. Sida caadiga ah, qiyaasta loogu talagalay dadka waaweyn waa 2 dhibcood oo ilaa 4 jeer maalintii. Iyadoo la tixgelinayo carruurta, xaddiga daroogada la go'aamiyo kaliya by dhakhtarka carruurta. Muddada aad daawada la dhibco lagu shubo indhaha iyo waa in lagu dhejiyaa uu dhakhtarka xaadirka ah.
Sida caadiga ah, muddada daawaynta qalab this waa wax ka badan 2 toddobaad. Laakiin haddii horumar lagu arkay, koorsada la soo kordhin karaa in ay muddo bil ah.
In kiiska lesions ballaaran xubnaha muuqaal ah oo halis ah, ka dibna dropwise Intaa waxaa dheer in irbado indhaha ah ay maamusho (diyaarinta beddelka ah).
Waayo, ka hortagga qalajiyo xuubka isha (halka ka shaqeeya computer a), waa in aad isticmaasho daawada 2 dhibcood inta lagu jiro maalinta la bareeg ah 2 saacadood.
waxyeellooyin
Waa maxay dhibaatooyinka daroogada waxay keeni kartaa "Thiotriazoline" (shots)? Tilmaamaha in habkan soo jeedisay in daawada si fiican loo dulqaatay si ixtiraam leh. Si kastaba ha ahaatee, iyadoo la isticmaalayo daroogada loo arkaa weli dhici karaan dareen diidmo oo aan loo baahnayn.
- nidaamka Central nervous: wareer, daciifnimo, dhaguhu dhegaha.
- mareenka dheefshiidka: afka oo qalala, lalabo, dibiro.
- Alaabteeda iyo wadnaha, cadaadiska dhiigga kor u kacay, tachycardia, arrhythmia, wadnaha xanuun.
- neefsashada, neefta iyo neefta oo ku qabata.
- Xasaasiyadda: qandho, dareen diidmo oo diidmo, anjioedema.
- reactions Local: casaan iyo dareen jidhidhico goobta la duray.
- falcelin maqaar: barrar maqaarka, cuncun, finan.
Sida dhibco lagu shubo indhaha, in ay ka qayb waxyeelo ah ayaa la arkay.
isdhexgalka daroogada
Sida laga soo xigtay khubaro, daroogada "Thiotriazoline" waxaa loo isticmaali karaa in lala daawooyinka aasaasiga ah ee loogu talagalay daaweynta cudurada wadnaha. Tan waxa u sabab xaqiiqada ah in ayaa sheegay in daroogada waa wakiilka ah cardioprotective.
Sidoo kale waa in la ogaadaa in daawada la oggol yahay in la isku mar lala isticmaalo daawooyinka lagu qoray daaweynta ku haboon ee hepatitis etiology.
Indhaha lagu dhibciyo "Thiotriazoline" ahaan loogu talo galay dumarka uurka leh iyo inta lagu jiro nuujinta. Waa in sidoo kale lagu sheegay in qaabka wax soo saarka ayaa sheegay in loo ogol yahay in ay isticmaalaan in lala siyaabo kale oo caafimaad.
Khamriga iyo Daroogada "Tiatriazolin" xoojin kasta oo kale ee ficil. Marka tan la eego, si ay u isticmaalaan saameen waa ka mamnuuc.
ganaaxyada
Walxaha ku jira kiniin sucrose tixgeliyo (qadarkuu of 2.8 mg kiniin). Sidaas darteed, si ay qiyaasta ugu badan ee maalin kasta daawada ku jiri kara oo ku saabsan 22,4 mg oo ah walaxda. Dhab ahaantii waxaa loo baahan yahay in la ogaado bukaanka, bukaanka qaba diabetes mellitus.
Hababka iyo caadada ee kaydinta
Absolutely dhammaan foomamka "Tiatriazolin" daroogada waa in laga ilaaliyo iftiin iyo meel aysan carruurta at heerkul ah 14 ilaa 26 digrii. Nolosha shelf ee daroogada waa 3 sano.
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