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Inhibitors Aromatase: dib u eegista, qiimaha. inhibitors Aromatase in bodybuilding

inhibitors Aromatase, ama blockers, - noocee ah ayuu bogsiinayay: qalab loo isticmaalo si loo yareeyo fiirsashada of estrogen ee dhiigga iyo in la kordhiyo heerka gonadotropins iyo testosterone. Waxyaabahani waxaa sidoo kale loo isticmaalaa daaweynta iyo ka hortagga gynecomastia lab.

inhibitors Aromatase in bodybuilding waxaa inta badan loo isticmaalaa inta lagu guda jiro koorsada ee steroids dhiska inay:

  • kor loogu qaado waxqabadka hormoonnada dhiska dhiigga;
  • ka hortagga gynecomastia;
  • looga hortago dhiig-karka,
  • kordhin bararto ah (by baabi'inta saamaynta xun ee estrogens);
  • yaraynta baabba 'estrogen dhidibka xiniinyaha-pituitary-hypothalamus taas oo horseedaysa in ay dib u dhiska degdeg ah,.

Dhisidda koorso, waa in aad xisaabtamin xaqiiqda ah in dhadhan ah oo aan ku xidhnayn oo dhan steroids dhiska. Isticmaal tahay waa laga caddeeyey markii isticmaalka waxa ka sameysan sida methandrostenolone, methyltestosterone, testosterone iyo taagayo ay. Wax yar ka dhadhan Halotestin, boldenone.

oolnimada

The inhibitors aromatase ugu doorbiday oo la heli karo, (waayo, Wax badan dhala ficil ahaan la mid ah):

article

(Title Global)

Brand (iibin by farmashiyayaasha)

qiimaha qiyaas

Form sii daayo

bodybuilding profilatikada

Marka gynecomastia ah

"Exemestane"

"AROMASIN"

1600 masaxo.

30 Tab. 25 mg

2.5 mg (kiniin bar) maalin kale oo kasta

25 mg maalin kasta ilaa iyo calaamadaha badanoo. Markaas qiyaasta yareynta in profilatikada.

'Letrozole'

"Letromara" (Farmak).

"Letroza"

"Estrolet"

3200 rubles.

1000 rubles.

30 Tab. 2.5 mg

0.5 mg (1/5 kiniin) maalin kale oo kasta

2.5 mg maalin kasta ilaa iyo calaamadaha reebay. Markaas qiyaasta yareynta si ka hortag ah.

"Anastrozole"

"Village"

"Egistrazol"

"Anastrozole Kabi"

1500 rubles.

350 rubles.

1300 masaxo.

28 Tab. 1 mg

0.5 mg (kiniin bar) maalin kale oo kasta

1 mg maalin kasta ilaa iyo calaamadaha badanoo. hoos dheeraad ah si ay qiyaasta profilatikada.

Waa in la ogaadaa in uruuray dhexdhexaad ah estrogen waa waxtar u leh koritaanka murqaha, qaadashada si kastaba ha ahaatee ka hortag tilmaamay in tiro saameeya ilaalinta ee heerka physiologically loo baahan yahay ee estrogens lab.

Isticmaalka koorsada

Inta badan ciyaartoyda gudaha isticmaalaya inhibitors aromatase, isticmaalaan xeeladaha soo socda: daroogada waxaa loo isticmaalaa oo kaliya marka calaamadaha ugu horeeya ee gynecomastia (cuncun ah ibta, barar, guduudasho). Nasiib darro, habkan ma la odhan karaa fiicnayn.

The xal ugu buuxa waxaa loo arkaa in lagu baaro estradiol in toban maalmood, isticmaalka steroids dhiska la bar-nolosha gaaban ( "Methandrostenolone", "propionate Hormoonkaas") ama saddex ama afar todobaad ee codsiga of Ester ee elongated ( "Sustanon", "enanthate," "cypionate"). Dheeraad ah oo ku qoray qayb celcelis "Anastrozole" - 0.5 mg maalin dhaaf. Toban maalmood ka dib, ku qabtay falanqayn gacanta of estradiol iyo qiyaasta la beddelo sida ay natiijada.

Tanaasulka waa in la isticmaalo inood u yar yahay oo dhexdhexaad ah "Anastrozole" diiradda on dareenkaa shakhsiyeed. Haddii ka dib markii daaweyn noocan oo kale ah uu noqonayaa mid niyadjab, disorder of function kacsi, dhibic libido, ka dibna aad u baahan tahay si loo yareeyo qiyaasta.

cilmi

ah ee a brand "letrazole" dadweynaha keenay wax soo saarka this hogaanka. Waxaa jira noocyo kala duwan oo baaritaan si loo caddeeyo oolnimada sare oo qalab this ragga. hordhaca ah ee walxaha ku weheliyay kor u calaamadeysan ee gonadotropin (LH). qiyaasta wax soo saar leh u billaabay ka 0.02 mg (daweyn hoos 100 jeer), waxaa suurto gal ah via saddexaad hoose fiirsashada estrogen ah. 50% "letrozole" jidhka ka reebtay 2-4 maalmood gudahood, jidaynayey inuu cabbo maalintii. khasaare aasaasiga ah waxaa loo arkaa inay awooddiisa ah inuu heerka hoose ee estrogen, xitaa in yar ka qaataan.

"Anastrozole" caanka ah ee bodybuilding, inuu cajiib bartay dadka iyada oo loo adeegsanayo yaraynta estradiol. Siman waxaa la muujiyey in qiyaas heerka estradiol 1-0.5 mg hoos u dhici doono ku dhowaad 50%. Ganacsatada wax soo saarka Tani ayaa laga soo iibsan karaa in ay toban jeer ka jaban tahay farmashiyaha. In megacities kulmay cheap "Anastrozole Kabi."

In uu buugga, Dr. Mauro G. De Pascal qoray: "Waxaa la qiyaasayo in estrogens in loo sameeyay iyadoo ay sabab u aromatization of testosterone ama steroids kale dhiska ee wasaaradaha ka mid ah hypothalamus iyo maskaxda, yaraynta dheecaan ka mid ah farabadan oo hormone, iyo, sidaas awgeed, wax soo saarka ee testosterone." Gilman iyo Goodman wargeliyay in warcelin waa halkii shaqeysiin raasamaal ah estrogen, halkii testosterone. Sidaas, waxaa la sheegay in ka inhibitors aromatase si weyn hoos ugu dhigi kartaa saamaynta inhibitory wakiilada dhiska loo qoondeeyo hormoonnada jinsiga shaqsi ah.

Dhibaatooyinka ay keento

The inhibitors aromatase ee khatarta ku ah dadka? Waxaan ognahay in estrogen ee qaadasho yar yahay waxay leeyihiin saamayn togan ku jidhka lab. hormoonnada Estrogen kordhiyo oo qiimeyn ku oolnimada iyo dareenka of receptors antiandrogen. Waxaa intaa dheer, iyagu leeyihiin saamayn difaaca iyo dhiska.

Taasoo la micno ah muruqa receptor estrogen si fiican ku tilmaamay in Anna Wiik si faahfaahsan. Dhab ahaantii dose xanibaha runtii cajiib ah loo baahneyn waxay yareyn kartaa heerka estrogen, kaas oo ku kordhinaya ah ee waxyeellooyin sida:

  • Iscelin of koritaanka murqaha;
  • kalagoysyada (arthralgia);
  • daraysa caafimaadka iyo hoos u dhac ku libido;
  • niyad-jabka,
  • disorder ee profile la egyahay dhiigga (cholesterol kordhay);
  • hoos u xoog lafaha.

Subjectively, daroogada waa dulqaadan badan "tamoxin".

inhibitors dabiiciga ah

Waa kuwan soo socda:

  • caffeine,
  • resveratrol;
  • zinc,
  • nicotine;
  • apigenin;
  • katychenz,
  • eriodiktiol.

Isticmaalka "Anastrozole"

In ka badan inhibitors aromatase wanaagsan? daawooyinkan hubkaas ayaa loo isticmaalaa in bodybuilding. Tusaale ahaan, "Anastrozole" looga baahan yahay haynta biyaha ee jirka aadanaha iyo ka hortagga dhacdo of gynecomastia (inta badan isku dhafan oo androgens testosterone iyo nooca Dianabol ama isku dhafan oo finasteride). Laakiin kiiskan, Orodyahanka helo oo ay la socdaan adag this cajiib ah daroogada mamnuuc ka ah "liiska walxaha laga mamnuucay iyo hababka", ka sokow isagoo ay kala duwan u gaar ah ee saamaynta sare.

Isticmaalka caasiyoobay ah ciyaartoyda "Anastrozole", ay qaadeen, gaar ahaan, bodybuilding keeni kartaa arthralgia, asthenia, ama in la yareeyo socodka ah ee laabatooyinka, madax-xanuun, somnolence. Dabcan, mararka qaar u muuqan kartaa dhibaato thromboembolic iyo horumarinta stroke.

On "Anastrozole" Wax badan ayaa laga qoray in suugaanta ee ciyaaraha fudud sida daroogada ah oo aad u dhib lahayn. Laakiin saamaynta fog oo deg deg ah ay ku soo dhaweynta waxay noqon kartaa mid aad u la saadaalin karin iyo naxdin leh. Indeed, haddii oo kaliya in ay qaataan hal kiniin (1 mg) maalin walba, la diyaarin karaa isxigxiga hormone dhawaaqaa. By habka, this ifafaale ayaa lagu arkay in ka badan 80% dadka loo isticmaalo wax soo saarka ah.

Guud ahaan, inhibitors aromatase - daroogada loo yaqaan ku filan. guud ahaan blockers baarka saddexaad "Anastrozole", oo mar dambe "vorozole" iyo
'Letrozole', la abuuray sida alaabta ka mid ah khadadka koowaad iyo labaad bogsiin kala firdhiyey kansarka naasaha receptor-positive.

"Krizin"

Waayo, weightlifters suuqa pharmacological sidoo kale bixisaa a 5.7-digidroksiflavon ( "Krizin"), taas oo ciyaartoyda isticmaalaan qaabab aad u sarreeya. Waxa uu ku antiaromatazatnymi oo la soo saaray ee laba nooc - MRM-Chrysin, jaan 500 mg halkii kaabsal krizina hufan iyo SciFit-Chrysin ES, jaan qeybtii walaxda firfircoon.

Dhibaatooyinka ay keento ku dhiirigelinayaan in uu ma uusan sheegin, laakiin waa in la xusuusto in dhammaan walxaha iyo diyaarinta isagoo talaabo antiaromatazatnym, wuxuu keeni karaa waxyeello jirka Orodyahanka cajiib ah. Intaas waxaa sii dheer, ay ku jiraan ee "List of walxaha mamnuuca ah iyo hababka."

Reviews

bodybuilders badan ayaa sheegaya in, ku salaysan waayo-aragnimo la "letrozole" ( "Femara"), waxay ku soo gabagabeeyey: Alaabta Tani, by xalinta mid dhibaato (tilmaame sare ee estrogen), kor u soo bixitaanka of dhibaatooyin kale oo badan. Dabcan, inhibitors aromatase ay muhiim u yihiin rag. Ka dib oo dhan, jidhka (ragga gaar ahaan) isticmaalaa estrogen si loo ilaaliyo caafimaadka ee habka difaaca jirka, maskaxda, heerka kolestaroolka caadiga ah, kala-goysyada caafimaad, seedaha, iyo wixii la mid ah.

Athletes sheegaya in estrogen ku kicin kara hab jirka ee koritaanka murqaha. Qaadashada 2.5 mg "letrozole" maalintii waxay bilaabaan inay dareemaan dhaawac halis ah goysyada articular iyo seedaha, oo noqday nugul cudurrada faafa iyo viral.

ciyaartoyda badan ayaa waxay aaminsan yihiin in 'Letrozole' waxaa loo isticmaali karaa oo kaliya bodybuilders xirfad loogu diyaar tartanka. Thanks isagii, ayay takhaluso dheecaanka dheeraadka ah ee jidhka (for xirfadlayaasha caafimaadka sababtoo ah guul ma aha xumahay). Waxay ku faraxsan yihiin in ay qaataan on inhibitor aromatase yihiin. Qiimahoodii waa arrin ku qanacsanayn.

ciyaartoyda Qaar waxay yidhaahdaan in saamayn togan 'Letrozole' on jidhka xitaa at dose oo ah 0.1-0.5 mg. Waxay sheegaan in ay tahay ma ka xun saamayn yar ee inhibitors kale, iyo heerka noocaan ah daawo. Waxay ku andacoodeen in subjectively, sheyga waxaa si deg deg revolutionizing mugga Testicular badan "tamoxin" iyo "Clomid". Waxay sidoo kale ku doodaya in ay inhibitors aromatase - daroogada in kharashka xaq tayo leh.

Qaar ka mid ah warbixin fudud loo isticmaali karo xanibaha kasta, laakiin marka la eego wax soo saarka sare "letrozole" ee qaadasho yar, waa kan ugu jaban.

"Anastrozole"

Maanta "Anastrozole" waa xanibaha ugu caansan. jaban ayaa loo arkaa ah "tuulada." Qaar ka mid ah inhibitors aromatase ee farmashiyaha waa dhif iyo naadir, tusaale ahaan, "Anastrozole Kabi."

Dad badan ma badbaadin on caafimaadkooda iyo dooran tayada.

Qaado "Anastrozole" si waafaqsan heerka gaarka ah ee estradiol. heerarka estradiol Sidaa darteed marka hore tijaabiyo si ay ula qabsadaan ku salaysan qayb falanqaynta. qiyaasta classical celcelis ahaan waa 0.5 mg maalintii.

Toban maalmood ka dib, waxaad u baahan tahay in mar kale la tijaabiyey. Haddii heerka estradiol heer, waxaa suurtagal ah si loo yareeyo qiyaasta ee 0.5 mg laba jeer toddobaadkii. Haddii weli waa sare, soo dhoweynta waa in la sii. Oo sidaas daraaddeed waxay noqon waa dhaqangaleyso illaa heer estradiol kabashada buuxda.

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