Caafimaadka, Diyaarinta
"Excedrin": dhigooda. daawo ee xanuunka dhanjafka "Excedrin": faallooyinka, qiimaha, analogs
Dhanjaf - taasi waa cudurka, taas oo aan la wareejin karaa iyada oo aan analgesics. Weerarka ayaa waxa uu awoodaa in uu socon muddo 4 maalmood ah. Ninka in muddo this lumiyo awoodda in ay ka shaqeeyaan. Isla mar ahaantaana uu isticmaalo daawo xoog leh in laga takhaluso xanuunsan dikaan wata ka. Laakiin, nasiib daro, ugu of qalab ah in la baabi'iyo karaa raaxo sida, qabatimo oo keeni xaqiiqada ah in cudurka uu noqdo chronic. Farmashiiste Modern ayaa sameeyay a daroogada cusub weyn. Means, iyo sidoo kale in laga takhaluso xanuunka dhanjafka, yaraynta awood u leh inay shaqeeyaan, laakiin ma aha in la qabatimo, daroogada waa "Excedrin". Analogs daroogada aan ka yarayn waa wax ku ool ah.
Sharaxaad kooban oo ku saabsan
daawo ee xanuunka dhanjafka "Excedrin" waa diyaarinta a weheliso tirsan kooxda analgesics-antipyretics. Waxa loo isticmaalaa madax xanuun aad u daran. Si tayo leh waxaa loola jeedaa "Excedrin" ka jaf. Xaaladdan oo kale, oo waxa uu xitaa ka hortagi kara weerarka.
Halabuurka The daroogada
waxtarka daawada ee been in waxyaabaha ay. daawada wuxuu ka kooban yahay:
- acetylsalicylic acid,
- caffeine,
- paracetamol.
Waa in walxahaasi mahad leedahay dhibaato kala duwan ee jirka ah. Sidaas darteed, balan qaadayo si degdeg ah, xanuun si buuxda u soo xirtey.
Paracetamol qadarkuu of 250 mg, Acetylsalicylic acid - 250 mg, iyo caffeine - 65 mg hal kiniin waxa ku jira daawooyinka "Excedrin". Halabuurka The sidaas, taasina waxay ka dhigan tahay sinji waa mid aad u muhiim ah. Sidaa darteed waxaa lagu talinayaa in la isticmaalo daroogada si taxadar leh u daran. Bukaan-socodka waa in ay tixgeliyaan qiyaasta ma badnayn.
Intaa waxaa dheer, daroogada waxaa ka mid ah maaddooyinka kaabayaal ah:
- giproloza;
- cellulose mikrokristallin;
- stearic acid.
Saamaynta ay jidhka
Kiniiniyada xanuunka dhanjafka "Excedrin" saddex qalab kala duwan oo ay leeyihiin guryaha kala duwan lagu sameeyo. Waxay isku dhafan oo u ogolaanaya in laga takhaluso xanuunka nooca kasta. Tan iyo dhanjafku ku weheliyay raaxo dheer iyo aad u daran, in laga takhaluso isaga waa in ay ahaadaan daawada aad u xoog badan. sida Taasi waa daroogada "Excedrin".
Maxaa qalab this ayaa sidoo kale ka hadlay saamaynta iyo saameynta? Jawaabta su'aasha been saamaynta on jirka ah ee qayb kasta oo ku jira daroogada:
- Paracetamol. walax waxay leedahay guryaha anti-bararka iyo qandho jabis ka xoogbadan. Waa inay awoodaan inay saamayn xarunta maskaxda in mas'uul ka yahay loo xakameeyo heerkulka ee hypothalamus ah. door muhiim ah ka tirtiridda dhanjafka waxa uu leeyahay tayo anti-bararka, maxaa yeelay, qandho uusan iska leh astaamaha cudurka.
- Acetylsalicylic acid. Qayb ka duwan guryaha qandhada fahmayaan. Eebe waa kan kara si aad yarayso oo baabi'iyo caabuq. In this yaraynaysaa xanuunka. Acetylsalicylic acid hortagi karaa dhacdo ee xinjiro dhiig. Waxaa istaago geedi socodka ka mid ah formation heerka gacanta, si fiican u wanaajisaa wareegga dhiigga ee meelaha barar ah.
- Caffeine. Doorka walax si ay u yareeyaan xanuunka ugu weyn. Aspirin iyo paracetamol ku meel gaar ah loo baabi'iyo karaa raaxo. Caffeine leedahay saamayn togan ku saabsan wareegga dhiigga ee maskaxda iyo waxay ka caawisaa laga takhaluso oo ka mid ah sababaha keena cudurkan. Waxaa intaa dheer, waxa ay u dareen neefsashada iyo xarumaha vasomotor, kor u ballaarinta marinnada dhiigga ee cidhiidhiga, ka hortagtaa xinjirowga ku qabanaya. Caffeine waa Fayda fiican daal iyo hurdo. Waxaa si weyn u kordhiyaa tayada oo ka mid ah u shaqeeyo iyo midab, Kuna horumarinta caafimaadka guud ee bukaan-socodka. isku dhafan ee aspirin la maalkii awood u hagaajinta socodka dhiigga oo si togan u saamayn weelasha maskaxda.
Heley taas diyaarinta waxaa laga codsadaa
Waxaa lagu talinayaa in la isticmaalo kiniinka "Excedrin" for syndromes xanuun ee adag fudud iyo kuwa dhexdhexaadka ah ee asal ahaan kala duwan:
- xanuunka dhanjafka,
- madax-xanuun,
- neuralgia,
- kedisa;
- myalgia, arthralgia (raaxo ee xubnaha iyo muruqyada);
- algomenorrhea (xanuunka caadada);
- syndrome xumad.
Pharmacokinetics
Xaaladaha intooda badan, daawada jirka "Excedrin" macquul ah si fiican loo dulqaatay. dib u eegista Consumer si buuxda loo xaqiijiyo this. saamayn noocan oo kale ah oo daroogada ah ayaa loo baahan yahay ee qaybaha:
- Paracetamol waa si fiican u nuugo in mareenka caloosha iyo mindhicirka. Waxaa la metabolized beerka, kelyaha iyo raaca sida glucuronide iyo sulfate conjugates. In ka yar 5% oo ka mid ah laga baxo wax qaab ah unmodified. Tan iyo bond protein plasma waa qiimo lahayn marka la isticmaalayo qiyaas caadiga ah daweynta. Laakiin iyadoo la kordhiyo in dambaysta ah - waxaa sii kordhaya. metabolite Hydroxylated sameeyay in tiro yar oo beer sarkhaansan oxidases isku qasan oo sida caadiga ah ay noqoto mid dhexdhexaad by qabanaya inay hiddo, ururto laga yaabaa in la badinta ah paracetamol oo keeni dhaawaca beerka.
- Acetylsalicylic acid si buuxda iyo si degdeg ah nuugo. Waxaa la hydrolyzed in dheefshiidka mareenka, dhiig iyo beerka. In foomka salicylates this. Dheeraad ah, ay metabolized beerka.
- Caffeine waxaa sidoo kale si degdeg ah si buuxda u nuugo. fiirsashada ugu badan ee jirka ku jira ayaa lagu arkay for 5-90 daqiiqo ka dib loo isticmaalin lacagaha calool madhan. Digo dhacaa sabab u ah Dheef-cagaarshowga. walax waxaa loo qaybiyey oo dhan dheecaannada jidhka. Isgaarsiinta la protein plasma waa 35%. Qeybta si buuxda loo metabolized iyo saxarrada kelyaha.
mudada kacmaha
Habboon ee maamulka afka ka dhigan tahay "Excedrin". Daawada waxaa loo isticmaalaa inta lagu guda jiro ama cuntada ka dib. Waxaa lagu talinayaa in ay biyo ka cabbaan ee u tiro badan.
dose Single ee dadka waaweyn iyo dhalinyarada (15 sano) - waa 1 kiniin saac oo kasta 4-6. Haddii qof uu dareensan yahay calaamadaha xanuunka dhanjafka ah aaddan, waxaa lagu talinayaa in la isticmaalo mar 2 kaniini. Tani waxay ka hortagi doonaan weerar xanuun. Si kastaba ha ahaatee, waa in mid ka mid ah la xasuusto in baabbi'iyee badan 6 unug maalintii gebi ahaanba la mamnuucay.
digniin muhiim ah
daawo wax ku ool ah waxaa loo ogol yahay in aad dalbato raaxo daran 3 maalmood. Inta lagu jiro wakhtigan, bukaanka waa in dhakhtarkaaga, kuwaas oo dooran doona habka kale oo kaamil ah by kuwaas oo si ay ula dagaalamaan cudurka la tasho.
Xaaladaha qaarkood, bukaanka waxaa lagu talinayaa in la kordhiyo isticmaalka daroogada. Laakiin go'aan noocan oo kale ah la sameeyo waxaa laga yaabaa in ku salaysan tilmaamo ku haboon oo kaliya dhakhtar takhasus u leh. Cun kiniiniga xanuunka dhanjafka "Excedrin" leedahay in ka badan 3 maalmood laguma talinayo. Kordhinta qiyaasta wuxuu keeni karaa cawaaqib xun. Sida dhaawaca beerka sabab u raasamaal ee metabolites ee jirka.
waxyeellooyin
Isticmaalka daroogada run ahaantii ma ku yeelan karaan saamayn wanaagsan ku jidhka. Tan iyo markii uu leeyahay tiro ka mid ah waxyeelo ka dhigan tahay "Excedrin". analogues Drug talin karaa daaweynta dhakhtarka, haddii aan daawada kor ku xusan waxaa haboon in bukaanka.
Sidaas daraaddeed, dhibaatooyinka soo socda:
- lalabo, matag,
- gastralgia;
- hepatotoxicity;
- lesions caloosha erosive iyo kolit;
- nephrotoxicity;
- cadaanyo;
- cadaadis sii kordhaya;
- tachycardia;
- wareer;
- bronchospasm;
- madax-xanuun,
- aragti cawlan,
- hoos ku xulkii dhiig xinjirowga sameeya ;
- tinnitus,
- dhiigbaxa syndrome (dhiig ciridka, goror, purpura);
- erythema malignant exudative (ama Stevens-Johnson syndrome);
- dhagihiisu culusyihiin,
- necrolysis sun epidermal (ama Lyell ee syndrome);
- cudurka kelyaha (Chance galleeyda papillary);
- horumarinta carruurta Raynaud ee syndrome (hyperpyrexia, aysiidh dheefshiidka, cudurada of habka dareemayaasha jirka iyo soo gunaanadeen, matag, beerka aan caadi ahayn).
Sababo in la helo
Nasiib darro, daawo ma noqon doonto mid wax ku ool ah oo loogu talagalay dadka oo dhan. Ka dib markii hab uu leeyahay tiro ka mid ah sababo. Waxay hubin in la tixgeliyo ka hor inta codsanaya. Laakiin quusan haddii daawada umana yimaado oo aan kharashka. dhakhtarka xaadirka ah waa mid aad u fududahay in la badalo qalab "Excedrin". Analogs oggolaadaan in la gaaro natiijo aan la aqbali karo.
Daawada waa u ee heley iyo shuruudaha soo socda:
- Diidmo in Cuntadan;
- boogaha caloosha iyo mindhicirka in marxaladda ba'an,
- neefta bronki,
- dhiigbaxa caloosha iyo mindhicirka,
- polyposis soo noq sanka (JQSHM paranasal);
- -diid si ay u NSAIDs;
- qalliin in raaco dhiigga,
- diathesis hemorrhagic,
- hypertension,
- hemophilia;
- gipoprotrombinemii;
- hypertension portal;
- glaucoma,
- ischemia daran wadnaha;
- K beriberi;
- la'aanta dehydrogenase glucose-6-phosphate,
- renal failure;
- uurka;
- nuujinta,
- hurdo xumo,
- caro;
- da'da carruurta ee (daroogada ma khuseeyo 15 sano).
xad dhaafka ah ee daawada
Daawo "Excedrin" dhanjafka waa in kaliya la qaataa qaabab kor ku xusan. Tan iyo wakiilka xadgudub keeni kartaa in dad badan oo la calaamadaha xun.
About xad dhaafka ah ee paracetamol tilmaamaya sifooyinka soo socda:
- Inta lagu jiro maalintii ugu horraysay waxaa caddaan maqaarka, matag, yalaalugo, calool xanuun, dheef glucose oo yaraada, anorexia, aysiidh dheefshiidka.
- 12-48 saacadaha shaqada ka dib markii jira astaamo ay suurtogal tahay beerka ka muujiyay la horumarka ee encephalopathy. Waayo, mid aad u daran oo xad dhaafka ah ee suuragalka ah - kooma iyo dhimasho. Waxaa laga yaabaa in kelyaha, Ulasocto galleeyda embriyaha, ganaca, arrhythmia.
Iska badinta xanaajiyeen by acetylsalicylic acid, waxay leedahay calaamadaha soo socda:
- Fudud - matag, yalaalugo, dawakhaad, aragga indhaha oo isku darsamay, tinnitus, madax xanuun.
- In lagu sumoobo daran - neefta oo ku qabata, dhiigrooraan, dyspnea, dhididka qabow dhegdheg, aysiidh neefsashada, curyaannimo neefsashada.
Xadgudubka sababa caffeine waxaa lagu qeexay by calaamadaha soo socda:
- gastralgia;
- cadhoodaan, walaaca,
- wareer;
- Xasillooni darro,
- fuuqbaxa;
- arrhythmia;
- kaadida oo soo noqnoqda,
- tachycardia;
- hyperthermia;
- kor u xanuun iyo dareen,
- gariirka,
- dhaguhu dhegaha,
- lalabo, matag (oo mararka qaarkood la joogitaanka dhiig);
- suuxdintu.
Haddii xad dhaafka ah waa in gargaar caafimaad oo degdeg ah. Intii lagu guda jiray 4 saacadood ee ugu horeeya waxaa lagu talinayaa in maydho caloosha, u abaari matag. Calool waa in la wada baabbe'een oo macnaheedu yahay "carbon kacsan".
analogues daawo
Xusuusnow in daroogo kasta waa in uu dhakhtarku soo qoro, tan iyo wakiilka kasta uu leeyahay tilmaamo iyo sababo ay.
Oo kaliya dhakhtar waa inay awoodaan inay ku bedelato daawo kale daroogada "Excedrin". Analogs of qayb hadda sida soo socota:
- "Akvatsitramon".
- "Atsifein".
- "Askofen".
- "Lagu daray Kofitsil."
- "Tsitramarin".
- "Migrenol dheeraad ah."
- "Tsitramon".
- "Tsitrapar".
Qiimaha daroogada
Wixii oo dhan ay wax ku-oolnimada, kharashka daawada aan qaali ahayn si ay macaamiisha "Excedrin" ka jaf. Price of baakadda (10 kiniin) kala duwan ee kala duwan ee 120-150 rubles. Qiimaha diyaarinta 20 kaniiniga of 210-250 rubles.
Isdhexgalka daawooyin kale
Bukaan-socodka qaata daawada "Excedrin" waa in la fahamsan yahay in kor loogu qaado karaan saamaynta on jidhka siyaabo kale sida:
- "Heparin";
- Daawada xinjirowga aan toos ahayn,
- "Reserpine";
- daroogada hypoglycemic;
- hormoonnada steroid.
Ogsoonow in isticmaalka isku mar lacagaha "Excedrin" la NSAIDs kale waxay keeni kartaa waxyeelo. Tusaale ahaan, in la dhexgalo daroogada protivopodagricakih, daroogada antihypertensive, waxay ka dhigan tahay "Furosemide" keenaysaa in hufnaan ku yar oo ka mid ah kooxaha daroogada.
opinion macaamiisha
daroogo kasta leeyahay (ma laga reebo iyo fayoobi "Excedrin") jawaabaha, labada togan iyo kuwa taban.
macaamiisha qaar ka mid ah daacad ah u sheegi, isagoo daroogada isku dayay mar, qayb iyaga la maayo. Dumar badan waa qalab wax ku ool ah in iyada kiishad. ma garan kartid marka weerarka xanuunka idin soo gaadhi doonaan. bukaanka noocan oo kale aragto in hal kiniin saacad awood u baabi'iyo calaamadaha xun. Iyo in ay dhacdo jaf daran meesha kaniiniyada daawada xanuunka 2 "Excedrin". Responses tilmaamaya oolnimada in aad u fiican oo ah qalab.
macaamiisha kale qaban dhibic kala duwan ee aragtida, odhanaya wax matare ka mid ah daroogada. Waxay ku doodayaan in walxaha firfircoon daawooyinka si gaar ah waxa laga iibsan karaa uga jaban tahay farmashiyaha. Si kastaba ha ahaatee, macaamiisha, kuwaas oo iloobin in ay noqon wax ku ool ah daroogada ahaa sabab u ah isku darka saxda ah ee dhammaan qaybaha in kasta oo kale oo la dhamaystiro si fiican.
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