Caafimaadka, Diyaarinta
"Pentoxifylline": analogues, tilmaamaha loo isticmaalo, qiimaha dhabta ah
Daawada waxaa lagu beddeli karaa by "Pentoxifylline?" analoogga ah daroogada loo soo bandhigi doonaa in qalabka maqaalka. ka waxaad ku baran doontaa waxa loola jeedo ayaa sheegay in foomamka medicament kuwaas oo waxaa la iibiyo, sida ay tahay in loo isticmaalo, iyo wixii la mid ah.
The Halabuurka, qaabka, baakadaha
In waxa foomka lagu iibiyo daawada "Pentoxifylline?" Tilmaamaha loogu isticmaalo (analogues daroogada this waxaa laga heli karaa farmashiye kasta) waxay muujinaysaa in daawada lagu heli karaa qaabab kala duwan, kuwaas oo:
- In kiniiniyada (400 iyo 100 mg) waxaa lagu dahaarka leh pink. In mid ka mid ah kartoonka ku jiri kara 60 ama 20 xabbo.
- kaabsal The (400 iyo 100 mg). pack The audio baakado laga yaabaa in 60 ama 20 xabbo.
- In kiniin, tallaabada dheer (600 iyo 400 mg) waxaa lagu dahaarka leh iyo enteric-dahaarka leeyihiin line a tahay horyaalka. kartoonka Baakadaha badaana wuxuu ka koobanyahay 50 gogo '.
- The fijaan oo xal loogu duray. Halabuurka ee dejinta waxaa ka mid ah pentoxifylline iyo sodium chloride iyo biyo.
Tilmaamo pharmacological
Waa maxay hantida ma daroogada "Pentoxifylline?" Analoogga ee hab this leedahay sifooyinka la mid ah sida medicament oo keliya ayaa sheegay in. Waxaa iska leh a lacag cusub group hemorheological pharmacological. Inuu awoodo inuu soo celiyo plasticity ee unugyada dhiigga cas iyo yareeyaan calaamadaha lahayo. Tani waxay kordhisaa permeability ee xididdada dhiigga, kaas oo ay leeyihiin Lumen cidhiidhi ah.
guryaha daroogada keenaysaa in microcirculation hagaagay, saamayn togan ku hypoxia unugyada.
Sidee "Pentoxifylline?" Analogues ee soo dejinta iyo Ruush leedahay saameyn la mid ah daweynta sida in lacagaha laftiisa. Ka dib isticmaalka daroogada, waxa ay yaraynaysaa xulkii of erythrocytes oo markii dambe si fudud loo kordhiyo socodka dhiigga xubnaha iyo dhex gelin galay jihada extravascular.
Waxaan ma dhihi karo in daawada loo arkaa yaraynaysaa nafwaayay dhiigga, sidaas kor u disaggregation dhiig xinjirowga. Sidaas darteed of saamaynta daroogada waa sii korodhay daqiiqo iyo stroke mugga, laakiin ma beddelo tirooyinka garaaca wadnaha.
Sayidka, weel ballaarinta sambabada hagaajinaysaa O 2 content dhiigga, iyo ballaarinta halbowleyaasha wadnaha in la kordhiyo O 2 bixinta si myocardium ah.
dejinta viewed awood sii kordhaysa ohyahay murqaha neefsashada iyo diaphragm. Under saameynta ay ku kordhinaysaa qadarka dhiigga ah ee dhex qulqulaya damaanadda, iyo sidoo kale socodka dhiigga wanaajiyey iyaga oo ku.
Waa maxay qaababka kale ee daroogada ayaa "Pentoxifylline?" Analoogga ee daroogada iyo daroogo laftiisa kordhin fiirsashada ee ATP ee maskaxda iyo in ay horumariyaan dhiigga gobollada ay waxyeello (tus, in stroke ischaemic) ah.
Sidoo kale waa in la ogaadaa in daroogada ayaa sheegay in ay saameyn wanaagsan ku habdhiska dhexe iyo hawlgalka. In lesions ee halbowlayaasha durugsan la isticmaalayo taasi ka dhigan tahay raadad si loo kordhiyo in masaafo socod, oo ay ku jiraan cudurro sida endarteritis obliterative.
beegyada uu pharmacokinetic
daroogada "Pentoxifylline" Muddo intee le'eg barbaro? Tilmaamaha loogu isticmaalo (analogues of dawadan hoos ku qoran) uu inoo sheegayaa in daroogada this awood u leeyahay in cabaar ah u fiican, oo ay ku jiraan iyada oo caqabad dhiig-maskaxda.
The bar-nolosha ee daroogada marka intravenously maamula waa 30 daqiiqo. Marka la helo daroogada waxaa gudaha si buuxda u nuugo ka soo mareenka caloosha iyo mindhicirka.
Medicament bedelay beerka, halkaas oo u yeela metabolites theobromine. The fiirsashada dhiigga ugu badan ee daroogada waxaa lagu gaarayaa 4 saacadood ka dib codsiga gudahood. Si kastaba ha ahaatee, waxa weli heer-daweynta ku saabsan maalin.
medicament soo bandhigay in kelyaha (qiyaastii 95%). xiidmaha dhex daawo baxay wax yar.
At jinsi ah caddaallad ah kan naaska, daroogada lagu sii daayo oo ay la socdaan caano ah. Sidoo kale waa in la ogaadaa in tirtiridda daroogada Kobocii in bukaanka qaba cudurka kelyaha ba'an, beerka iyo dadka waayeelka ah.
Tilmaamayaasha loo isticmaalo
Waayo, waa maxay ujeedada bukaanka ahaan loogu talo galay dawada "Pentoxifylline?" Analogs iyo keydka daroogada waxay leeyihiin tilmaamo mid ah.
Currently, sida daroogada wax ku ool ah waxaa loo isticmaalaa in lagu daaweeyo cudurro badan. Halkan haatana waxa ay yihiin:
- deficiency cerebrovascular;
- urolithiasis,
- encephalopathy arteriosclerotic;
- stroke ischaemic;
- nefroangiopatiya diabetic;
- hypertension,
- boronkiitada obstructive;
- neefta bronki,
- xanuunada wareegga dhiigga durugsan ;
- encephalopathy;
- algomenorrhea;
- sepsis;
- cholecystitis,
- Tardive xiidmaha ;
- pilorospazm;
- adkaashada murqaha siman,
- post-trombophlebitic syndrome,
- dysmenorrhea;
- angioneyropatii (cudur Raynaud ee) ;
- xanuunada wareegga dhiigga indhaha,
- cudurada unugyada trophic;
- boogaha trophic;
- halis dhicin,
- cudurada functional of dhexe iyo dhegta gudaha;
- impotence vascular,
- Dystrophy muruqa;
- gangrene, qadhqadhyo.
sababo
Waa kuwee cudurada waxaa ka mamnuuc ah isticmaalka daroogada "Pentoxifylline?" analoogga ah oo ka mid ah daroogada iyo daroogo laftiisa in aan loo qaadan karaa dadka qaba dulqaad in qaybaha ugu muhiimsan, iyo sidoo kale wakiillo kale oo ka tirsan kooxda xanthine ah.
Intaa waxaa dheer, daroogada loo arkaa ahaan uu u bukaanka qaba dhawaan soo gaaray a stroke dhiigbaxa ama Wadnaxanuun myocardial ba'an iyo sidoo kale ka cabanaya atherosclerosis qalbiga daran iyo xididdada maskaxda, porfyri.
isticmaalka daroogada xididka waxaa reebban arrhythmia, dhiigbaxa, cadaadiska dhiigga oo hooseeya, hemorrhages in ileyska. Sidoo kale, daroogada waa u inta lagu jiro nuujinta iyo uurka, carruurta jirta ilaa 18 sano.
Iyadoo taxadar gaar ah ayaa loo diraa waxay ka dhigan tahay dadka ku shaqeeya (si looga hortago dhiig ee xub-axaleedka iyo xubnaha gudaha), iyo dadka qaba kelyaha ba'an iyo beerka, cudurka boog xiidmaha, gastritis iyo wadnaha oo shaqadiisa gaba.
Hababka Isticmaalka
Sida loo isticmaalo daroogada "Pentoxifylline?" Tilmaamaha loogu isticmaalo, dhabta ah (analogues qalab this laga yaabaa in qaadashada kala duwan) dhakhaatiirta la kulantay ayaa sheegaya in daroogada taas waxaa loo hadal iyo parenterally qaaday (ku xiran tahay darnaanta cudurka).
Maamulka Oral daroogada bilowdo dose oo ah 200 mg (i.e., 2 kaniini sadex jeer maalintii, cuntada ka dib). Ka dib markaad gaartey tirada cayiman saamaynta ku daweynta waa la dhimay by badh. Koorsada kaniiniyada daawada waa in aan ka badnayn hal bil socon.
In cudurro xunxun oo ba'an ee xubnaha gudaha daawo maamula in kaabsulka. Waxaa jira 2 siyaabood oo ka mid ah maamulka daroogada, xididka iyo intraarterial. Habka ugu horeysay ay fuliyeen walax ah. Waayo, kanu Ujeedada, 1 weelka 250 ml xal glucose ama chloride sodium. qiyaasta ayuu yiri waxaa maamula 2 saacadood gudahood.
Sida maamulka intraarterial, waxaa la maamulo ee dose oo ah 0.1 g halkii 50 ml of xal sodium chloride.
waxyeellooyin
Waxaa ka mid ah dhibaatooyinka ugu badan waa kuwa soo socda:
- wareer, welwel, hurdo xumo, qalal, isbedel dabeecadda qofka, madax-xanuun,
- daridda cholecystitis, transaminases beerka kacsantahay, horumarinta hepatitis cholestatic;
- matag, dareen ee buuxnaanta caloosha, yaqyaqsi, shuban ah, rabitaanka cuntada oo luma;
- finan, shoog, cuncun, barar angioneurotic, casaan maqaarka,
- dhacdo ee garaaca, wadnaha xanuun, hoos u cadaadiska dhiigga, stenokardicheskie xanuun;
- Torombositobiiniya, leukopenia;
- hoy, arag isku darsan;
- daridda xiiqda, bronchospasm, yaridu neefsashada;
- dhiig ee etiology kala duwan.
Drug "Pentoxifylline": analogues, qiimaha
Analogs waxaa loo arkaa daawooyinka dawooyinka soo socda:
- dragees "Agapurin" (100 mg) oo xal la isku duro ee ampoules (100 mg);
- kiniiniyada "Pot", kiniinada (600 mg);
- dragees, kiniin iyo xal isku duro "Trental".
Waa in la ogaadaa in "Trental" ka dhigan tahay daroogo asalka ah. Wuxuu waxa lagu qoray bukaanka qaba encephalopathy asal ahaan kala duwan.
Sida qiimaha, ka dibna diyaarinta oo dhan waa kala duwan yahay. Analoogga "Trental" "Pentoxifylline" waxa laga iibsan karaa 120 rubles medicament asalka ah - 520 rubles "Agapurin" - 300 rubles, halka "Pot" - 400 rubles.
Reviews
Reviews ku saabsan daroogada tani waa inta badan wanaagsan. Daawada waa wax ku ool ah ee cudurrada vascular xubnaha iyo nidaamyo badan. dib u eegista Inta badan ee ku saabsan isticmaalka "Pentoxifylline" ay ka soo tageen nin la ildaran xaaqyna endarteritis la claudication go'aysa. medicament Tani waa iyaga u adeegsanayo № 1, tan iyo markii cudurka tani waxay noqonaysaa inay horumar.
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