CaafimaadkaDiyaarinta

"Buspirone": dib u eegista, tilmaamaha loo isticmaalo, analogs

"Buspirone" waxaa loola jeedaa lacagta in ay leeyihiin saamayn on habka dareemayaasha jirka. Waa anxiolytic, loogu talagalay in lagu baabi'iyo welwel iyo cabsi, caadi hurdo, wanaajiyo fayo-qabka ay goobjoog ka ahaayeen neurosis. Kiniiniga "Buspirone" waa sababo qaar ka mid ah, oo keeni kartaa waxyeelo.

The Halabuurka iyo qaab "Buspirone" daroogada

Daawada waxaa laga heli karaa qaab kiniin ah ee qiyaasta a of 5, 10 iyo 20 mg. The walax daroogada firfircoon - buspirone. walxaha darran waxaa ka mid ah hydroxide potassium, galleyda, milmahayn magnesium.

saamaynta pharmacological

tallaabo ee ku dejinaysaa daroogada, anxiolytic. Daawada ka saaraysaa calaamadaha cabsi of daaqsinka iyo caafimaadka maskaxda. macnaheedu waa hab ay of action waxaa si buuxda ma ay garan, laakiin waxaa la ogsoon yahay in "Buspirone" waa ka benzodiazepines iyo daroogooyinka kale saamayn anxiolytic kala duwan.

A saamayn xoog inhibitory on yimaada habdhiska dhimirka ka dib markii la helo looxyadii offline "buspirone". Tilmaamaha loogu isticmaalo muujinaysaa in daroogada ay yaraynaysaa dhismaha iyo sii daayo serotonin, gaabisaa serotonergic, kor u dopamine xanibeen D2-receptors (boosteejada postsynaptic iyo presynaptic), dedejisaa excitation ee neurons dopamine ku yaalla maskax-ka. Ka dib markii la baabiiyo of daroogada aan arkay dhacdo ee astaamaha u-barashada iyo walaaca soo laabtay.

Daawada waxaa loogu tala galay maamulka afka. Cabaar galay jidhka in muddo gaaban markii uu si buuxda u nuugo jirta marinka dheef shiidka. Sidaas darteed, dheef ballaaran bioavailability waa keliya 4%. Heerka ugu badan ee daroogada ee dhiiggiisa la soo gaadhay oo ku saabsan saacad ka dib markii lays geliyey mareenka caloosha iyo mindhicirka. Half-nolosha waxaa lagu fuliyaa 2-3 saacadood, ku qabanaya borotiinka plasma u dhiganta 95%. isticmaalka joogtada ah "buspirone" wax saameyn ah kuma ay ku oolnimada.

Inta lagu jiro daaweynta, ma kaliya filan ee "Buspirone" waxaa loola jeedaa saamayn. Tilmaamaha loogu isticmaalo muujinaysaa in waxtarka daawada waa in muddada u dhaxaysa 7-dii ilaa maalinta 14-ka mid ah uu ogolaado. Saamaynta ugu badan ee daroogada ku muujiyey oo ku saabsan 120 maalmood ee daaweynta ka dib.

Tilmaamayaasha "buspirone"

Khubarada qoro dawooyinka marka dareensan khatarta, daaha ka cabsi iyo walwal, ee ma suuroowdaa jid caro dhiirogelin ka dhaca neurosis iyo hurdo xanuunada sahlan, kaas oo ay leeyihiin qof nidaamsan. Shayga haboon daaweynta xanuunada degaaankaaga, dystonia daaqsinka iyo niyad-jabka waa, la baabi'iyo stress, khamriga.

Sababo in la helo "Buspirone" daroogada

"Buspirone" (analogues daroogada iyo sidoo) ayaa sababo. daroogada asalka reebay in ay qaataan in kiisaska noocaas ah:

  • glaucoma (nooca xiran);
  • geeddi socodka bahal culus dhaca beerka iyo kelyaha,
  • qalalka,
  • xanuunada wadnaha, dhibaato xididdada dhiigga,
  • lesions of mareenka-mareenka,
  • daweeyay gravis;
  • Diidmo in qaybaha ah;
  • xilliga dhalmada, dabiibayo uu xabadka;
  • da'da ka yar 18 sano.

Haddii ay jirto waa mamnuuc in ay u qoraan dadka kiniiniga in a "Buspirone" bukaanka taariikh suuxitaan ama qalalka.

Ka hor inta aadan bilaabin daawaynta waa inay hubiyaan dareenka bukaanka ee daroogada.

Isticmaalka lacagta, qiyaasta

Inta lagu guda jiro daawaynta ka dhigan tahay "buspirone" codsiga kaniiniyada ka dhigay si waafaqsan talooyinka dhakhtarka daaweynta. guide rasmiga ah ku qoran warbixin in loo baahan yahay, waayo, mid kasta oo qiyaas kala duwan ee bukaanka, ie. circuit daaweynta Individual K. go'aamisa waxtarka therapy sameeyaa. qiyaasta waxay ku xiran tahay caafimaadka bukaan-socodka. talooyinka guud waa sida soo socota:

  • stage horudhac ah - 3 qiyaasood oo ah 5 mg ah ee daawada,
  • sii therapy - korodh ah ee dose waafaqsan bareeg ka mid ah 2-3 maalmood (haddii ay jirto baahi noocan oo kale ah);
  • maamulka qiyaas badnaan maalin kasta of 50 mg (ay ka maqan yihiin saamaynta doonay).

Kiniiniga tilmaamaha "Buspirone" loo isticmaalo ogolaanshaha qaadan oo keliya qaab guud ahaan, ma ay la kala diri karaa in dareeraha ah, sicir- oo calaliyo. Dawadu waa ku sakhraamin xaddi, mudda oo biyo ah, qaato waqti kasta oo ah maalintii madax banaan cunto qaadashada. Muddada heerka lagu taliyey in 4 bilood. The dheer waqtigan loola dhaqmo "buspirone" laguma talinayo.

Waxyeellada "buspirone"

Marka daaweynta daroogada qaar ka mid ah falcelinta aan loo baahnayn ee u shaqeeyo waxaa lagu ogaan karaa. Tusaale ahaan, la qabsi, daraysa caafimaadka guud, daciifnimo, daal, arxandarro. Haddii ay jiraan saamaynta sida waxay u baahan tahay ka saarida daroogada. Waa in la xiriir dhakhtarka iyo isaga wargeliyo oo ka mid ah isbedel xun ee jirka ka dib qaadashada kiniinka "Buspirone". Tilmaamaha loogu isticmaalo kiisaska noocaas ah waxaa lagu talinayaa in la dhimo cadadka wakiilka. Haddii waxyeelo kaa tagi waayaan, dhakhtarku wuxuu leeyahay si uu u bedelo daroogooyinka kale daawo dheeraad ah oo ku haboon.

Mararka aad dhif u ah, isticmaalka "buspirone" keenaysaa in rabshooyin ee habka dheef shiidka. Tusaale ahaan, waxaa laga yaabaa in lallabo iyo laab, raaceen by matag. xanuun suurto gal ah in gobolka gaastari. Waxaa laga yaabaa in waxyeelo kale. calaamadaha Oo intaas oo dhammu waxay muujinayaan dulqaad ka mid ah qaybaha daroogada.

Iska badinta "Buspirone" daroogada

Haddii qalab loo isticmaalo qaabab ka badan talinayaa, qofka la kulmi karaan astaamaha badinta. Waxaa ka mid ah lalabo iyo matag, xanuunada caloosha ah nooc kale. wareer The bukaanka, gaabiso ardayda, waxay noqon kartaa khasaare kooban oo miyir. Bukaan-socodka tago dib u eegis daaweynta ka dib waxaa loola jeedaa "Buspirone Sandoz", ayaa xusay suurtagalnimada ee qasnaanta, gariirka ee qeybta sare. Ka mid ah daliilka kale ee xad dhaafka ah - caro, caro, Isbedellada joogtada ah ee niyadda. Overdosing waxaa lagu daaweeyaa by lavage gastric, maamulka carbon shaqeysiin ee jirka, daaweynta calaamadaha iyo qabashada gacanta joogta ah cadaadiska dhiigga, garaaca wadnaha, dhaqdhaqaaqa neefsashada. daawo u gaar ah gargaarka ee calaamadaha ah qiyaasta xad dhaafka "buspirone" kajirin. Dialysis xaaladahan oo kale ma keeni saamaynta doonayo.

Dhexgalka walxaha kala duwan iyo daroogooyinka kale

Mararka qaarkood marka la isku daray mamnuuc daawooyin gaar ah kaniiniga tilmaamaha "Buspirone" loo isticmaalo ee analogues ku talinaysaa in ka fiirsaneysa inuu bedel u yahay xarunta asalka ah. Waxaa la og yahay in daawada waa in aan la isku soo qaaday la dajiye, daawada dajiyaha ay sabab u tahay kor loogu qaado saamaynta daawooyinka laga qaado. In daaweynta "buspirone" loo baahan yahay in laga saaro isticmaalka cabitaanka khamriga. Waxaad ma isku dari kartaa daawada la MAO sababtoo ah khatarta ah ee dhibaatada hypertensive.

Marka aad isticmaali labada "Haloperidol" with "buspirone" dhiigga ku kordhiyaa heerka daroogada this. Isku darka daawada la "trazodone" keenaysaa in koror weyn oo ALT.

Sidaas darteed of tijaabo ku lug leh xoolaha, Saameynta xun ee u shaqeeyo aan la ogaado inta lagu jiro daaweynta. Si kastaba ha ahaatee, si looga fogaado dareen diidmo oo aan loo baahnayn oo jidhka ah in ay aqbalaan waa in la siiyo.

tilmaamaha "Buspirone" si loogu isticmaalo waa sida qalab kuwaas shiid beerka. In nidaamka this ka qayb CYP3A4, isagoo isoenzyme qayb diyaarinta shaqeeyo processing. Sababtan awgeed, xidhiidhka ka dhici kara "buspirone" daawooyin kuwaas oo inducers, ama inhibitors ee eulayska.

Features of isticmaalka daroogada

Haddii, inta lagu jiro nuujinta, waxaa loo baahan yahay therapy, oo ku salaysan soo dhoweynta ee "buspirone" naas-meel gaar ah joojin.

Waxaa jira qaar ka mid ah xayiraad marka carqalad ah shaqaynaya ee xubnaha gudaha. Tusaale ahaan, haddii aad qabto dhibaatooyin beerka waa inay ka taxadiraan inta lagu jiro muddada daawaynta oo si joogto ah loola socdo isbedelada ka dhaca caafimaadka. Sababo kaliya aan caadi ahayn daran dhaxgalka ee jirka. Isla sidaas u dhaqmaan shaqo ee kelyaha.

Ku saabsan magacaabidda wakiilada ka saarayaasha kala duwan, in H. Vol. "Buspirone Sandoz" daroogada, dib u eegista caafimaadka soo jeedin baahida loo qabo in ay ixtiraamaan sharciyada qaarkood. Qoraalka ka soo daawada, takhasus u leh waa inay ogaadaan in qalab this ma awoodo inuu baabi'iyo astaamaha ka dhalanaya ka Benzodiazepin, iyo ujeedada xaaladahan oo kale suurtogal ma aha, haddii aan xirxirin daroogada anxiolytic la soo saaray ka hor inta therapy ah.

Bukaan-socodka waa in ay ogaadaan in kaniiniyada "Buspirone" saamayn ku yeelan kara daryeelka, gaar ahaan bilowga hore ee daaweynta, sidaa daraadeed waxa fiican in si ku meel gaar ka fogaadaan hawlaha ku lug leh mas'uuliyad gaar ah iyo ka-fiirsashada kordhay. Qaar ka mid ah hawlaha uu noqon karaa mid khatar ku ah caafimaadka.

Iyadoo la tixgelinayo therapy ee macnihiisu yahay "Buspirone", dhakhaatiirta dhab ah oo ku saabsan daroogada oo inta badan wanaagsan. Si kastaba ha ahaatee, khubarada tilmaamay in ay lagama maarmaan tahay in ay ku wareejiso si sax ah oo kaliya la tilmaamo ku haboon iyo in qiyaasood oo aan fiicnayn. Waa in la ogaadaa in walwalka iyo walaaca ka kici ka saameynta joogtada ah negative walaaca maalin kasta, daaweynta la anxiolytics badanaa muhiim ma aha.

Aqbaliddoodii ka dhigan tahay bukaanka "buspirone" la qiyaasta kala duwan, tus daroogo "buspirone 10 mg" ratings wakiil isticmaalka hab wax ku ool ah. Dadka ayaa lagu daaweeyo daawo this, la soco in dhakhtar uu uga digay in ay isticmaalka taxadir daawooyinka qaarkood, sida kaniinka ka hortaga, daawooyinka sonkorowga, wakiilada in bar hoos u cadaadiska dhiigga ee sareeya, daroogada in la baabi'iyo murugada iyo daawooyin sida glycosides wadnaha , neuroleptics.

kelyaha iyo beerka cirrhosis daran u baahan hoos cutubyo qiyaasta. Xaaladahan, habka of "Buspirone Sandoz" dib u sida dadka ku tilmaami daaweynta in loo baahan yahay in loo maamulo iyada oo ay kormeerayaan dhakhtar. Ogaanno waxaa lagu sawiray isbedelka yar ee caafimaadka.

Bukaanka qaba daawooyinka qalalka marnaba qoray, maxaa yeelay, khatarta ah qalal. daaweynta noocan oo kale ah dadka bukaanka ah waa khatar ah iyo waa in la fuliyaa iyadoo la isticmaalayo daawooyinka kale. Bukaanka inta badan xadgudbo daawooyinka iyo waxay leeyihiin taariikh ah oo ku tiirsanaanta daroogada waa in la daaweeyaa iyada oo ay kormeerayaan adag ee takhasus leh (dhacdooyinka ku xiran "buspirone" ma ahaa).

Daraasado ayaa muujiyey in "Buspirone" 3-4 toddobaad daaweynta ka dib marka alarm ma aha wax ku ool ah, sidaas darteed ma jiro dareen in iyaga lagu daweeyo muddo dheer. Sababo la helid la'aanta macluumaad ku saabsan ammaanka daroogada in carruurta uu ballan looma samayn in qof ka yar da'da 18 sano.

Daaweynta kala duwanaansho kala duwan ee "hexane Buspirone" daroogada iyo daawada dib u khubarada qaar ayaa tilmaamaya sida therapy xumaada sabab ah in seexan dhibaatooyin, soo bixitaanka of caro iyo walaac mararka qaar waa calaamad ka mid ah xanuunada psychomotor halis ah.

Analogs, dib u eegista ku saabsan "Buspirone" daroogada

analog daroogada bedelka waa in la sameeyaa ka dib helitaanka talo dhakhtar. Waxaa jira bedel u fiican tahay daawo, "Buspirone" - "Spitomin". Kurtumm muujiyaan in ay talaabo la mid tahay tallaabo oo ka mid ah lacagta asalka ah. "Spitomin" waxaa loo isticmaalaa daaweynta kuwa xaaladaha lagu cabudhibayo iyo "Buspirone". Reviews waa wanaagsan yihiin, sidaas darteed haddii aad u baahan tahay in ay suuragal tahay in ay ka faa'iidaystaan bedel this, laakiin kaliya ka dib markii uu la tashado takhasus u leh. Saameyn la mid ah waxaa lagu gaarayaa ay sabab u tahay jiritaanka qayb ka mid ah oo firfircoon. The "Spitomin" ugu waxtarka badan ayaa muujinaya in daaweynta bukaannada qaba jirrada walaaca.

daawaynta ka dib markii Kurtumm "Buspirone" tagi karo kala duwan, laakiin asal ahaan natiijada daaweynta sida waa ay wanaagsan tahay. Ma xaqiijiyay ay waxtarka? Reviews dhakhtarro ayaa tilmaamaya in wax soo saarka la hydrochloride buspirone qayb firfircoon waa la si guul la diriraya daliilka walaaca kala duwanaan karaan darnaanta iyo asal ahaan, laakiin ay saamayn mar shiidaa dareemo, waxa loo arki karaa oo kaliya waqti cayiman ka dib, kuwaas oo - hal ama laba todobaad ka dib. Si aad u aragto saameyn ku daweyn suurto gal ugu badan, waxay u baahan yihiin in la daweeyo muddo hal bil ah.

"Buspirone" helo jawaabo wanaagsan bukaannada ku jira xaaladaha halkaas oo ma jiraan waxyeelo, oo uu daroogada niyad jabka wanaagsan. Mararka qaarkood waxaa jiri doona falcelin xun ee u shaqeeyo, laakiin aad u dhif ah marka jirku uusan ogayn qaybaha daroogada. Laga soo bilaabo dib u eegista ah, waxa ogaaday in daaweynta waxaa la socon kara by teraabiyada cilminafsiga iyo hawlaha sotsioterapevticheskimi. Marmarka qaarkood bukaanka waxay leeyihiin dhibaato caloosha iyo mindhicirka, wareer iyo daciifnimo. Iska badinta - ifafaale dhif ah.

Sidaas darteed, isticmaalka daroogada jawaabaha "Buspirone" bukaanka loola dhaqmo Dabcan, dhif tago macluumaad ku saabsan saameyn khatar ah. Dabcan waa in ku salaysan sifooyinka gaarka ah ee jidhka bini'aadamka, caafimaadkiisa, oo aan fiicnayn, waayo, kiis kasta qaadasho. In kasta oo ay gacanta ku joogto dhakhtarka, bukaanka waxaa looga baahan yahay in uu akhriyo tilmaamaha inta aadan bilaabin daaweynta.

"Buspirone" - daroogada ah in inta badan laguma keeni horumarinta dhibaalka dhanka kale iyo badinta, non-qabatin leh, horumarka xun ka dib markii ay la joojiyo, oo kiisaska intooda badan ma ay shaqo.

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